Buy N-Methyl-Cyclazodone now
N-Methyl-Cyclazodone is an approximately 2x – 4x more potent derivative of the nootropic and psychostimulant compound Pemoline.
|Form||White or off-white powder|
|Molecular Weight||230.26 g/mol|
|Synonyms||N-Cyclopropyl-N-Methylpemoline, 2-(Cyclopropyl(methyl)amino)-5-phenyl-2-oxazolin-4-one, 2-(Cyclopropyl(methyl)amino)-5-phenyloxazol-4(5H)-one, LD 4202|
N-Methyl-Cyclazodone provided particularly strong central stimulant and motor excitant properties, such that a dose of 1 mg/kg in the mouse proved the compound to be equal in potency to d-amphetamine, but longer lasting in effect. The anorexigenic effect of the compound was also similar to that of d-amphetamine; however, unlike d-amphetamine, the compound was not a convulsant, had substantially lower toxicity, and had only a very slight cardiovascular effect in doses up to 5 mg/kg parenterally in the cat or dog.
N-Methyl-Cyclazodone is an N,N-disubstituted pemoline derivative. As an N,N-disubstituted compound, the literature indicates that Thozalinone shows milder and less potent, but potentially more sustained stimulant and antidepressant effects than N-monoalkyl pemoline derivatives. By analogy, this could suggest the possibility that the pharmacological effects of N-Methyl-Cyclazodone could be slightly milder and less potent, but longer lasting than those of Cyclazodone. Also likely as a result of N,N-disubstitution, the patents disclosed that N-Methyl-Cyclazodone (in comparison to Cyclazodone) had a comparatively lower melting point of 94-95°C.